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Pharmacology and Toxicology

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Showing page 9 of 22 pages of list content

  • Validation and invalidation of SARS-CoV-2 papain-like protease inhibitors

    This article's authors
    1. Chunlong Ma
    2. Jun Wang
    This article has 1 evaluations Latest evaluation on Nov 19, 2021 Published on Nov 5, 2021
  • Brilacidin, a COVID-19 Drug Candidate, demonstrates broad-spectrum antiviral activity against human coronaviruses OC43, 229E and NL63 through targeting both the virus and the host cell

    This article's authors
    1. Yanmei Hu
    2. Hyunil Jo
    3. William F. DeGrado
    4. Jun Wang
    This article has 1 evaluations Latest evaluation on Nov 19, 2021 Published on Nov 5, 2021
  • Novel pectin from crude polysaccharide of Syzygium aromaticum against SARS-CoV-2 activities by targeting 3CLpro

    This article's authors
    1. Can Jin
    2. Bo Feng
    3. Rongjuan Pei
    4. Yaqi Ding
    5. Meixia Li
    6. Xia Chen
    7. Zhenyun Du
    8. Yangxiao Ding
    9. Chunfan Huang
    10. Bo Zhang
    11. Xinwen Chen
    12. Yi Zang
    13. Jia Li
    14. Kan Ding
    This article has 1 evaluations Latest evaluation on Nov 19, 2021 Published on Oct 29, 2021
  • Characterization of raloxifene as potential pharmacological agent against SARS-CoV-2 and its variants

    This article's authors
    1. Daniela Iaconis
    2. Carmine Talarico
    3. Candida Manelfi
    4. Maria Candida Cesta
    5. Mara Zippoli
    6. Francesca Caccuri
    7. Giulia Matusali
    8. Licia Bordi
    9. Laura Scorzolini
    10. Enrico Bucci
    11. Arnaldo Caruso
    12. Emanuele Nicastri
    13. Marcello Allegretti
    14. Andrea Rosario Beccari
    This article has 1 evaluations Latest evaluation on Nov 19, 2021 Published on Oct 24, 2021
  • μ-Theraphotoxin-Pn3a inhibition of CaV3.3 channels reveals a novel isoform-selective drug binding site

    This article's authors
    1. Jeffrey R. McArthur
    2. Jierong Wen
    3. Andrew Hung
    4. Rocio K. Finol-Urdaneta
    5. David J. Adams
    This article has 4 evaluations Latest evaluation on Nov 15, 2021 Published on Oct 4, 2021
  • Characterization of the Endogenous DAF-12 Ligand and Its Use as an Anthelmintic Agent inStrongyloides stercoralis

    This article's authors
    1. Zhu Wang
    2. Mi Cheong Cheong
    3. Jet Tsien
    4. Heping Deng
    5. Tian Qin
    6. Jonathan D. C. Stoltzfus
    7. Tegegn G. Jaleta
    8. Xinshe Li
    9. James B. Lok
    10. Steven A. Kliewer
    11. David J. Mangelsdorf
    This article has 4 evaluations Latest evaluation on Nov 12, 2021 Published on Sep 8, 2021
  • Covalent inhibition of endoplasmic reticulum chaperone GRP78 disconnects the transduction of ER stress signals to inflammation and lipid accumulation in diet-induced obese mice

    This article's authors
    1. Dan Luo
    2. Ni Fan
    3. Xiuying Zhang
    4. Fung Yin Ngo
    5. Jia Zhao
    6. Wei Zhao
    7. Min Huang
    8. Ding Li
    9. Yu Wang
    10. Jianhui Rong
    This article has 4 evaluations Latest evaluation on Nov 10, 2021 Published on Aug 20, 2021
  • Predicting drug polypharmacology from cell morphology readouts using variational autoencoder latent space arithmetic

    This article's authors
    1. Yuen Ler Chow
    2. Shantanu Singh
    3. Anne E. Carpenter
    4. Gregory P. Way
    This article has 8 evaluations Latest evaluation on Nov 7, 2021 Published on Sep 3, 2021
  • Bisphosphonate drugs have actions outside the skeleton and inhibit the mevalonate pathway in alveolar macrophages

    This article's authors
    1. Marcia A. Munoz
    2. Emma K. Fletcher
    3. Oliver P. Skinner
    4. Julie Jurczyluk
    5. Esther Kristianto
    6. Mark P. Hodson
    7. Shuting Sun
    8. Frank H. Ebetino
    9. David R. Croucher
    10. Philip M. Hansbro
    11. Jacqueline R. Center
    12. Michael J. Rogers
    This article has 5 evaluations Latest evaluation on Nov 1, 2021 Published on Aug 10, 2021
  • Repurposed nystatin to inhibit SARS-CoV-2 and mutants in the GI tract

    This article's authors
    1. Eszter Virág
    2. Dénes Seffer
    3. Ágota Pénzes-Hűvös
    4. Krisztina Varajti
    5. Géza Hegedűs
    6. István Jankovics
    7. József Péter Pallos
    This article has 1 evaluations Latest evaluation on Oct 23, 2021 Published on Oct 20, 2021
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